1 |
ICV371 |
36.27 | 73.22% | 49.54% |
virus: Papain-like protease; 3C-like protease | P0DTD1 | SARS 3CL(IC50=30.2µM); MERS 3CL(IC50=34.7µM); MERS PL(IC50=48.8µM) |
2 |
ICV276 |
32.31 | 70.96% | 45.53% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=6.1µM) |
3 |
ICV299 |
31.66 | 70.19% | 45.11% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=5µM) |
4 |
ICV372 |
30.74 | 69.44% | 44.26% |
virus: Papain-like protease; 3C-like protease | P0DTD1 | SARS 3CL(IC50=84.8µM); MERS PL(IC50=88.5µM) |
5 |
ICV275 |
30.42 | 66.28% | 45.9% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=6.2µM) |
6 |
ICV374 |
29.96 | 70.41% | 42.55% |
virus: Papain-like protease; 3C-like protease | P0DTD1 | SARS 3CL(IC50=92.4µM); MERS 3CL(IC50=125.7µM); MERS PL(IC50=49.1µM) |
7 |
ICV280 |
29.66 | 71.38% | 41.55% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=9.2µM) |
8 |
ICV277 |
28.55 | 64.74% | 44.09% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=11.6µM) |
9 |
ICV279 |
27.95 | 68.7% | 40.69% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=9.5µM) |
10 |
ICV206 |
27.75 | 72.98% | 38.03% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(EC50=23µM) |
11 |
ICV282 |
27.4 | 67.24% | 40.74% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=12.7µM) |
12 |
ICV284 |
26.78 | 65.24% | 41.04% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=10.4µM) |
13 |
ICV286 |
26.68 | 72.78% | 36.67% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=7.8µM) |
14 |
ICV376 |
26.55 | 59% | 45% |
virus: Papain-like protease; 3C-like protease | P0DTD1 | SARS 3CL(IC50=64.2µM); MERS 3CL(IC50=109.2µM); MERS PL(IC50=55µM) |
15 |
ICV278 |
26.11 | 58.74% | 44.44% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=12.5µM) |
16 |
ICV288 |
26.03 | 63.9% | 40.74% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=12.3µM) |
17 |
ICV283 |
25.95 | 59.92% | 43.31% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=14.4µM) |
18 |
ICV285 |
25.58 | 64.64% | 39.57% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=13.9µM) |
19 |
ICV369 |
25.25 | 75.14% | 33.6% |
virus: Papain-like protease; 3C-like protease | P0DTD1 | SARS 3CL(IC50=202.7µM); MERS 3CL(IC50=193.7µM); MERS PL(IC50=171.6µM) |
20 |
ICV426 |
25.12 | 65.45% | 38.38% |
human: Estrogen receptor | P03372 | MERS(EC50=10.117µM) Vero E6; SARS(EC50=92.886µM) Vero E6 |