1 |
ICV256 |
15.41 | 79.63% | 19.35% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=2.25µM) |
2 |
ICV274 |
14.97 | 70.94% | 21.11% |
virus: Papain-like protease | P0DTD1 | MERS PL(IC50=20µM) |
3 |
ICV254 |
14.94 | 75.74% | 19.72% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=12.66µM) |
4 |
ICV261 |
14.85 | 80.34% | 18.49% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=13.86µM) |
5 |
ICV253 |
14.52 | 76.16% | 19.07% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=4.45µM) |
6 |
ICV255 |
14.52 | 76.48% | 18.98% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=1.18µM) |
7 |
ICV252 |
14.43 | 80.22% | 17.99% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=51.33µM) |
8 |
ICV250 |
14.4 | 76.93% | 18.72% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=34.91µM) |
9 |
ICV262 |
14.17 | 75.34% | 18.81% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=17.82µM) |
10 |
ICV260 |
13.84 | 70.82% | 19.55% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=9.91µM) |
11 |
ICV257 |
13.74 | 72.72% | 18.89% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=4.3µM) |
12 |
ICV141 |
13.48 | 73.21% | 18.41% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=39.87µM) |
13 |
ICV140 |
13.35 | 74.71% | 17.87% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=14µM) |
14 |
ICV177 |
13.35 | 72.93% | 18.3% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=4.3µM) |
15 |
ICV247 |
13.21 | 69.6% | 18.98% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=76.74µM) |
16 |
ICV176 |
13.21 | 67.08% | 19.69% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=0.31µM) |
17 |
ICV175 |
13.16 | 76.94% | 17.1% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=0.03µM) |
18 |
ICV136 |
12.79 | 71.57% | 17.87% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=1.04µM) |
19 |
ICV36 |
12.76 | 67.7% | 18.85% |
virus: 3C-like protease | P0DTD1 | MERS 3CL(IC50=6.7µM); SARS 3CL(IC50=10.9µM) |
20 |
ICV258 |
12.74 | 67.74% | 18.81% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=11.83µM) |