1 |
ICV392 |
23.16 | 61.77% | 37.5% |
virus: Helicase | P0DTD1 | SARS Helicase(IC50=5.4µM) |
2 |
ICV284 |
22.63 | 68.14% | 33.2% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=10.4µM) |
3 |
ICV373 |
21.57 | 61.98% | 34.8% |
virus: Papain-like protease; 3C-like protease | P0DTD1 | SARS 3CL(IC50=233.3µM); MERS PL(IC50=94.9µM) |
4 |
ICV285 |
21.3 | 63.4% | 33.59% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=13.9µM) |
5 |
ICV282 |
20.93 | 62.32% | 33.59% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=12.7µM) |
6 |
ICV72 |
20.92 | 69.42% | 30.13% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=2.5µM) |
7 |
ICV199 |
20.19 | 67.39% | 29.97% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=62.79µM) |
8 |
ICV280 |
20.09 | 62.34% | 32.22% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=9.2µM) |
9 |
ICV202 |
19.71 | 66.46% | 29.66% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=90.72µM) |
10 |
ICV372 |
19.37 | 59.05% | 32.8% |
virus: Papain-like protease; 3C-like protease | P0DTD1 | SARS 3CL(IC50=84.8µM); MERS PL(IC50=88.5µM) |
11 |
ICV281 |
19.33 | 58.21% | 33.21% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=13.2µM) |
12 |
ICV440 |
19.11 | 52.19% | 36.62% |
human: Synaptic Vesicular amine transporter | Q05940 | SARS(EC50=3.4µM) Vero E6 |
13 |
ICV276 |
19.08 | 65.02% | 29.34% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=6.1µM) |
14 |
ICV200 |
19.05 | 63.21% | 30.14% |
virus: 3C-like protease | P0DTD1 | SARS 3CL(IC50=101.38µM) |
15 |
ICV279 |
19.03 | 59.71% | 31.87% |
virus: Papain-like protease | P0DTD1 | SARS PL(IC50=9.5µM) |
16 |
ICV73 |
18.87 | 67.28% | 28.04% |
virus: 3C-like protease | P0DTD1 | Replicon (BHK) (IC50=2µM); SARS(IC50=8.9µM) Vero |
17 |
ICV428 |
18.41 | 58.75% | 31.34% |
human: Eukaryotic initiation factor 4A-I | P60842 | MERS(EC50=3nM) MRC-5 cell; HCoV-229E(EC50=1.3nM) MRC-5 cell |
18 |
ICV403 |
18.35 | 54.41% | 33.72% |
virus: Envelope protein; Spike protein | QHD43418.1,P0DTC2 | FIPV(EC50=7.8µM) Black TN406HP |
19 |
ICV374 |
18.27 | 57.56% | 31.73% |
virus: Papain-like protease; 3C-like protease | P0DTD1 | SARS 3CL(IC50=92.4µM); MERS 3CL(IC50=125.7µM); MERS PL(IC50=49.1µM) |
20 |
ICV390 |
18.21 | 65.42% | 27.84% |
virus: Helicase | P0DTD1 | SARS Helicase(IC50=7µM) |